発表論文

【2021 年】

54) Apocynin-tandospirone Derivatives Demonstrate Antioxidant Properties in the Animal Model of Schizophrenia
T. Uehara, M. Kurachi, T. Kondo, H. Abe, Q.-L. Zhao, H. Itoh, T. Sumiyoshi, M. Suzuki
Adv. Redox Res., 3, 100013 (2021). DOI: 10.1016/j.arres.2021.100013.

53) Synthesis of Nilotinin M3: An Ellagitannin Containing an Isodehydrodigalloyl Group
H. Imai,Y. Kanzaka, Y. Sunatsuki, H. Abe
Synthesis, 53, 3630-3638 (2021); DOI: 10.1055/a-1508-9541.

52) Total Synthesis of Urolithin C 3-Glucuronide
K. Itaya,I. Jeelani, H. Abe
Heterocycles, 103, 1038-1047 (2021).

51) Synthesis of Chloro-substituteed 6H-Dibenzo[b,d]pyran-6-one Natural Products, Graphislactone G, and Palmariols A and B
H. Abe, I. Jeelani, A. Yonoki, H. Imai, Y. Horino
Chem. Pharm. Bull, 69, 781-788 (2021).

50) Preparation of Isodehydrodigallic Acid Using Ullmann Condensation
H. Imai, R. Koyama, Y. Horino, H. Abe
Chem. Pharm. Bull., 69, 298-301 (2021).

49) Total Synthesis of Hyalodendriol C
I. Jeelani, K. Itaya, H. Abe
Heterocycles, 102, 1570-1578 (2021).


【2020 年】

48) 抗酸化機能を付与したハイブリッド型神経保護薬の創製
上原隆、倉知正佳、近藤隆、阿部仁、鈴木道雄
バイオインダストリー, 37 (7) , 29-40 (2020).

47) 抗酸化機能を付与したタンドスピロン誘導体−新規神経保護薬の創製
上原隆、阿部仁、倉知正佳、近藤隆、鈴木道雄
化学工業, 71, 298-305 (2020).

46) Synthesis of Lactonized Valoneoyl Group-containing Ellagitannins, Oenothein C and Cornusiin B
H. Abe, H. Imai, D. Ogura, Y. Horino
Heterocycles, 101, 524-535 (2020).

【2019 年】

45) DMSO-Perturbing Assay for Identifying Promiscuous Enzyme Inhibitors
K. Tomohara, I. Adachi, Y. Horino, H. Kesamaru, H. Abe, K. Suyama, T. Nose
ACS Med. Chem. Lett., 10, 923-928 (2019).

44) Anti-psychotic Drugs Scavenge Radiation-induced Hydroxyl Radicals and Intracellular ROS Formation, and Protect Apoptosis in Human Lymphoma U937 Cells
Q.-L. Zhao, H. Ito, T. Kondo, T. Uehara, M. Ikeda, H. Abe, J.-I. Saitoh, K. Noguchi, M. Suzuki, M. Kurachi
Free Radic. Res., 53, 304-312 (2019).

43) Trialkylborane-Mediated Multicomponent Reaction for the Diastereoselective Synthesis of Anti-,-Disubstituted Homoallylic Alcohols

Y. Horino, M. Murakami, A. Aimono, J. H. Lee, H. Abe
Org. Lett., 21, 476-480 (2019).

☆ 特願 2019-95359、タンドスピロン誘導体
近藤隆、阿部仁、倉知正佳、上原隆


【2018 年】

42) Total Synthesis of Coriariin B
H. Abe, Y. Kato, H. Imai, Y. Horino
Heterocycles, 97, 1237-1247 (2018).

【2017 年】

41) Controllable Stereoselective Synthesis of (Z)- and (E)- Homoallylic Alcohols Using a Palladium-Catalyzed Three-Component Reaction
Y. Horino, M. Sugata, I. Mutsuura, K. Tomohara, H. Abe
Org. Lett., 19, 5968-5971 (2017).

40) Improved Synthesis of Nigricanin
H. Abe, T. Nagai, H. Imai, Y. Horino
Chem. Pharm. Bull., 65, 1078-1080 (2017).

39) ビアリールカップリング反応を利用する天然物合成
阿部仁
有機合成化学協会誌, 75, 850-863 (2017).

38) Palladium-Catalyzed Diastereoselective Synthesis of Homoaldol Equivalent Products
Y. Horino, M. Sugata, T. Sugita, A. Aimono, H. Abe
Tetrahedron Lett., 58, 2131-2134 (2017).

37) Total Synthesis of Oenothein C
H. Abe, D. Ogura, Y. Horino
Heterocycles, 95, 131-136 (2017).


【2016 年】

36) Facile Synthesis of (Z)-anti-Homoallylic Alcohols from 3-(Pinacolatoboryl)allyl Alcohols, Aldehydes, and Triorganoboranes via a Palladium-Catalyzed Three-Component Reaction
Y. Horino, A. Aimono, N. Minoshima, H. Abe
Tetrahedron Lett., 57, 3561-3564 (2016).

35) Palladium-Catalyzed Three-Component Reaction of 3-(Tri-n-butylstannyl)allyl Acetates, Aldehydes, and Triorganoboranes: An Alternative to the Carbonyl Allylation Using α,γ-Substituted Allylic Tin Reagents
Y. Horino, M. Sugata, H. Abe

Adv. Synth. Catal., 358, 1023-1028 (2016).
Highlighted in Synfacts, 12, 611 (2016).

34) Initial Synthesis of Valoneic and Woodfordinic Acid Dilactones
H. Abe, S. Ishikura, Y. Horino
Synlett, 27, 859-863 (2016).

33) Synthesis of 2,3,9,10-Tetraoxygenated Benzo[c]phenanthridine Derivatives via Palladium-mediated Aryl-aryl Coupling Reaction
H. Abe, N. Kobayashi, Y. Kadoshima, Y. Takeuchi, T. Harayama, Y. Horino
Heterocycles, 93, 673-684 (2016).


【2015 年】

32) Palladium-catalyzed Three-Component Reaction of 3-(Pinacolatoboryl)ally Acetates, Aldehydes, and Organoboranes: A New Entry to Stereoselective Synthesis of (Z)-anti-Homoallylic Alcohols
Y. Horino, A. Aimono, H. Abe
Org. Lett., 17, 2824-2827 (2015).

31) Palladium-mediated Intramolecular Biaryl Coupling Reaction: Convenient Preparation of Furoquinolinone Derivatives
H. Abe, M. Kamimura, Y. Komatsu, Y. Horino
Heterocycles, 90, 1332-1342 (2015).


【2014 年】

30) Palladium-Catalyzed Cyclopropanation of Strained Alkenes with 3-Pinacolatoboryl-1-arylallyl Carboxylates
Y. Horino, Y. Takahashi, R. Kobayashi, H. Abe
Eur. J. Org. Chem.,7818-7822 (2014).

29) Practical and Convenient Synthesis of 1,6-Di- or 1,2,5,6-Tetra-arylhexa-1,3,5-trienes by the Dimerization of Pd(0)-Complexed Alkenylcarbenes Generated from π-Allylpalladium Intermediates
Y. Horino, Y. Takahashi, K. Koketsu, H. Abe, K. Tsuge
Org. Lett., 16, 3184-3187 (2014).

28) Regioselectivity of the Palladium-mediated Intramolecular Coupling Reacton of Highly Oxygenated Phenyl Benzoate Derivatives and Application to the Synthesis of Alternenuol
T. Matsukihira, S. Saga, Y. Horino, H. Abe
Heterocycles, 89, 59-68 (2014). 

27) Regioselectivity of the Intramolecular Biaryl Coupling Reaction of 3-Substituted Phenyl 2-Iodobenzoate Using a Palladium Reagent
K. Maeda, T. Matsukihira, S. Saga, Y. Takeuchi, T. Harayama, Y. Horino, H. Abe
Heterocycles, 88, 621-628 (2014).

26) Relay Catalysis Using a Gold(I) Complex/Bronsted Acid Binary System for the Synthesis of Benzoxasiloles
Y. Horino, Y. Takahashi, Y. Nakashima, H. Abe
RSC Adv., 4, 6215-6218 (2014).


【2013 年】

25) Facile Preparation of Dehydrodigallic Acid and Its Derivative for the Synthesis of Ellagitannin
K. Shioe, S. Ishikura, Y. Horino, H. Abe
Chem. Pharm. Bull., 61, 1308-1314 (2013).

24) Synthesis of Nigricanin via Intramolecular Biaryl Coupling Reaction of Fnctionalized Phenyl Benzoate
T. Matsukihira, T. Kida, K. Hidaka, S. Saga, M. Takemura, A. Yonoki, T. Nishimori, Y. Horino, T. Harayama, Y. Takeuchi, H. Abe
Heterocycles, 87, 2555-2565 (2013).


【2012 年】

23) Synthesis of Neo-tanshinlactone via the Palladium-mediated Intramolecular Biaryl Coupling Reaction

H. Abe, T. Kawai, Y. Komatsu, M. Kamimura, Y. Takeuchi, Y. Horino
Heterocycles, 86, 785-789 (2012).

22) Highly Regioselective Intramolecular Biaryl Coupling Reaction of a Phenyl Benzoate Derivative for the Synthesis of Graphislactone G
H. Abe, T. Matsukihira, T. Fukumoto, Y. Horino, Y. Takeuchi, T. Harayama
Heterocycles, 84, 323-326 (2012).


【2011 年】

21) Synthesis and Anti-human Immunodeficiency Virus Activity of the Skeleton Isomers of 3′,4′-Di-(O)-(−)-camphanoyl-(+)-khellactone
H. Nishioka, K. Uesugi, N. Ueda, Y. Kondo, M. Tsuji, H. Abe, T. Harayama, T. Hamasaki, M. Baba, Y. Takeuchi
Chem. Pharm. Bull., 59, 1075-1076 (2011).

20) Synthetic Studies of Substituted Pyridine Aldehydes as Intermediates for the Synthesis of Toddaquinoline, Its Derivatives and Other Natural Products
G. Serban, H. Abe, Y. Takeuchi
Heterocycles, 83, 1989-2000 (2011).

19) Synthesis of (-)-Actinonin
S. Inoue, H. Nishioka, H. Abe, T. Harayama, Y. Takeuchi
Synthesis, 1705-1710 (2011).

18) Syntheses of All-Methylated Ellagitannin, Isorugosin B and Rugosin B
K. Shioe, Y. Sahara, Y. Horino, T. Harayama, Y. Takeuchi, H. Abe
Tetrahedron, 67, 1960-1970 (2011).


【2010 年】

17) Synthesis of Acinetobactin
Y. Takeuchi, S. Ozaki, M. Satoh, K. Mimura, S. Hara, H. Abe, H. Nishioka, T. Harayama
Chem. Pharm. Bull., 58, 1552-1553 (2010).

16) Regioseletivity in Direct Arylation of Benzanilide Possessing Oxygen Substituents in the Benzoyl Part Using Palladium without Phosphine Ligand
T. Harayama, C. Nagura, T. Miyagoe, Y. Kawata, H. Abe, Y. Takeuchi
Heterocycles, 81, 2609-2616 (2010).

15) Reactions of Nonsymmetrical Bidentate Linkers Having a Phthalimidoyl and Acid Chloride Group or a 2-Benzothiazole Group with α-D-Glucoside Derivatives and Their Application for the Modification of Cellulose
M. C. Sheikh, S. Takagi, H. Abe, T. Yoshimura, H. Morita
Carbohydr. Res., 345, 2562-2565 (2010).

14) Synthesis of Graphislactone H
H. Abe, T. Fukumoto, Y. Horino, T. Harayama, Y. Takeuchi
Heterocycles, 82, 851-855 (2010).

13) Effect of Oxygen Substituent in the Aniline Part of Benzanilide on the Regioselectivity in Direct Arylation Using Palladium-phosphine Reagents
T. Harayama, M. Asai, T. Miyagoe, H. Abe, Y. Takeuchi, A. Yamaguchi, S. Fujii
Heterocycles, 81, 1881-1889 (2010).

12) Studies on the Lossen-type Rearrangement of N-(3-Phenylpropionyloxy)phthalimide and N-Tosyloxy Derivatives with Several Nucleophiles
M. C. Sheikh, S. Takagi, A. Ogasawara, M. Ohira, R. Miyatake, H. Abe, T. Yoshimura, H. Morita
Tetrahedron, 66, 2132-2140 (2010).

11) Synthesis of All-methylated Isorugosin B
K. Shioe, Y. Takeuchi, T. Harayama, H. Abe
Chem. Pharm. Bull., 58, 435-437 (2010).

10)  Synthesis of Zanthoxyline and Its Related Compounds: Revision of the Reported Structure
H. Abe, N. Kobayashi, Y. Takeuchi, T. Harayama
Heterocycles, 80, 873-877 (2010).


【2009 年】

9) Lossen-Type Rearrangement Products in the Reaction of N-(Phthalimidoyloxy)-3-phenylpropionate and -Tosylate with Benzyl Alcohol
S. Takagi, M. C. Sheikh, A. Ogasawara, M. Ohira, H. Abe, H. Morita
Heterocycles, 78, 1433-1438 (2009).

8) Preparation of 5H,7H-Dibenz[c,e]oxepin-5-one Derivative through Reconstruction of the Lactone Ring

H. Abe, M. Arai, Y. Takeuchi, T. Harayama

Heterocycles, 77, 1409-1416 (2009).


【2008 年】

7) First Synthesis of Non-symmetrical "Phthalimidoyl Active Ester" Bi-dentate Cross-linking Reagents Having an Acid Chloride, 2-Benzothiazole, or 1-Benzotriazol Group
M. C. Sheikh, S. Takagi, M. Sakai, H. Abe, H. Morita
Org. Biomol. Chem., 6, 4505-4508 (2008). 

6) Concise Asymmetric Synthesis of (+)-Febrifugine Utilizing trans-Selective Intramolecular Conjugate Addition

S. Sukemoto, M. Oshige, M. Sato, K. Mimura, H. Nishioka, H. Abe, T. Harayama, Y. Takeuchi

Synthesis, 3081-3087 (2008).

5) Generation of Nitrene by the Photolysis of N-Substituted Iminodibenzothiophene

H. Morita, A. Tatami, T. Maeda, B. J. Kim, W. Kawashima, T. Yoshimura, H. Abe, T. Akasaka

J. Org. Chem., 73, 7159-7163 (2008).

4) Synthesis of Highly Oxygenated Biphenyl Derivative in an Optically Active Form through Palladium-Mediated Intramolecular Biaryl Coupling Reaction

H. Abe, M. Arai, K. Nishioka, T. Kida, K. Shioe, Y. Takeuchi, T. Harayama

Heterocycles, 76, 291-303 (2008).

3) A New Approach to the Benzopyridoxepine Core by Metal Mediated Intramolecular Biaryl Ether Formation

G. Serban, H. Abe, Y. Takeuchi, T. Harayama

Heterocycles, 75, 2949-2958 (2008).

2) Palladium-Mediated Intramolecular Biaryl Coupling Reaction for Natural Product Synthesis

H. Abe, T. Harayama

Heterocycles, 75, 1305-1320 (2008).

1) Enantioselective Synthesis of Valoneic Acid Derivative

H. Abe, Y. Sahara, Y. Matsuzaki, Y. Takeuchi, T. Harayama

Tetrahedron Lett., 49, 605-609 (2008).

2007 年以前の論文はこちら  

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